BindingDB Entry 5280: S18616, a highly potent, spiroimidazoline agonist at alpha(2)-adrenoceptors: I. Receptor profile, antinociceptive and hypothermic actions in comparison with dexmedetomidine and clonidine.

BindingDB

Description

No description available.

Citations (0)

Mentions (0)

Metrics

Dataset Index

24.5

FAIR Score

52%

Citations

60

Mentions

0

Metrics Over Time

Publication Details

DOI

Publisher

BindingDB

License

Attribution 3.0 United States

Assigned Domain

Subfield

Molecular Biology

Field

Biochemistry, Genetics and Molecular Biology

Domain

Life Sciences

Confidence Score

100%

Source

Open Alex

Keywords

Adrenergic alpha1B, Adrenergic receptor alpha, Alpha adrenergic receptor 1A and 1B, Alpha-1A adrenergic receptor, Alpha-1D adrenergic receptor, Alpha-2A adrenergic receptor, Alpha-2B adrenergic receptor, Alpha-2C adrenergic receptor, Beta-1 adrenergic receptor, Beta-2 adrenergic receptor and beta-3 adrenergic receptor, Imidazoline I1, Monoamine Oxidase Type B (MAO-B), Monoamine oxidase, Sodium-dependent noradrenaline transporter, and adrenergic Alpha2, Centre de Recherches de Croissy, Affinity

Normalization Factors

FT

53.85

CTw

1.00

MTw

1.00