Published on 01 January 2010

BindingDB Entry 50031502: Discovery and optimization of 2-(4-substituted-pyrrolo[2,3-b]pyridin-3-yl)methylene-4-hydroxybenzofuran-3(2H)-ones as potent and selective ATP-competitive inhibitors of the mammalian target of rapamycin (mTOR).

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Description

No description available.

Citations (0)

Mentions (0)

Metrics

Dataset Index

0.3

FAIR Score

13%

Citations

0

Mentions

0

Metrics Over Time

Publication Details

DOI

Publisher

BindingDB

Assigned Domain

Subfield

Molecular Biology

Field

Biochemistry, Genetics and Molecular Biology

Domain

Life Sciences

Confidence Score

69%

Source

Scholar Data Model

Keywords

Aurora kinase B/Inner centromere protein, Cyclin-dependent kinase 1, Cyclin-dependent kinase 2, Fibroblast growth factor receptor 1, Glycogen synthase kinase-3, Hepatocyte growth factor receptor, Inhibitor of NF-kappa-B kinase (IKK), MAP kinase ERK2, MAP kinase-activated protein kinase 2, Mitogen-activated protein kinase 14, Mitogen-activated protein kinase 2, PI3-kinase subunit alpha, Platelet-derived growth factor receptor, Protein kinase C alpha type, Rho-associated protein kinase, Ribosomal protein S6 kinase alpha 1, SRC, Serine/threonine-protein kinase mTOR, Tyrosine-protein kinase ABL1, VEGF-receptor 2 and tyrosine-protein kinase SRC, and Vascular endothelial growth factor receptor 2, Wyeth Research, Affinity

Normalization Factors

FT

13.46

CTw

1.00

MTw

1.00