BindingDB Entry 50043836: Discovery of 1-methyl-1H-imidazole derivatives as potent Jak2 inhibitors.
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Publication Details
Subfield
Molecular Biology
Field
Biochemistry, Genetics and Molecular Biology
Domain
Life Sciences
Confidence Score
68%
Source
Scholar Data Model
Keywords
ALK tyrosine kinase receptor, Casein Kinase II, Casein kinase II, Fibroblast growth factor receptor 1, Focal adhesion kinase 1/vascular endothelial growth factor receptor 3, JAK3/JAK1, Kinesin-1 heavy chain/ Tyrosine-protein kinase receptor RET, LIM domain kinase 1, Neurotrophic tyrosine kinase receptor, Non-receptor tyrosine-protein kinase TYK2, Protein kinase C (PKC), SRC, Serine/threonine-protein kinase Aurora, Serine/threonine-protein kinase SIK1, Tyrosine-protein kinase ABL1, Tyrosine-protein kinase JAK1, Tyrosine-protein kinase JAK2, Tyrosine-protein kinase JAK3, Tyrosine-protein kinase receptor FLT3, and Vascular endothelial growth factor receptor 2, AstraZeneca, Affinity