Published on 01 January 2020
BindingDB Entry 50005393: Discovery of potent selective bioavailable phosphodiesterase 2 (PDE2) inhibitors active in an osteoarthritis pain model. Part II: optimization studies and demonstration of in vivo efficacy.
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Publication Details
Subfield
Molecular Biology
Field
Biochemistry, Genetics and Molecular Biology
Domain
Life Sciences
Confidence Score
71%
Source
Scholar Data Model
Keywords
3',5'-cyclic phosphodiesterase and Homo sapiens phosphodiesterase 2A (PDE2A), Pfizer Inc., Affinity